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Medicinal Chemistry
ISSN: 1573-4064 - Volume 4, 6 Issues, 2008

Editor-in-Chief:
Atta-ur-Rahman, FRS
HEJ Research Institute of Chemistry
University of Karachi
Karachi - 75270
Pakistan
Co-Editors:
Andreas Hilgeroth
Martin-Luther-Universitaet Halle-Wittenberg
Halle
Germany
William J. Hoekstra
Viamet Pharmaceuticals
Durham, NC
USA
Associate Editors:
K.C. Chou (Gordon Life Science Institute,
San Diego, USA)
I.A. McDonald (Pharmaxis Ltd., Frenchs Forest, Australia)
H. Kalasz (Semmelweis University, Budapest, Hungary)
D.M. Lambert (Catholic University of Louvain, Brussels,
Belgium)
I. Toth (University of Queensland, Brisbane, Australia)
Editorial Advisory Board:
S.S. Abdel-Meguid (Delta Search
Labs, MA, USA)
T. Abe (Medicinal Chemistry Research Lab,
Yokohama, Japan)
W-R. Abraham (German Research Centre for
Biotechnology, Braunschweig, Germany)
S. Ahmed (Kingston University, Thames Surrey,
UK)
R. Andersen (British Columbia, Vancouver,
Canada)
V. Apostolopoulos (The Austin Research Institute,
Heidelberg, Australia)
S. Balaz (North Dakota State University,
Fargo, USA)
A. Balkan (Hocettepe University, Ankara,
Turkey)
P.G. Baraldi (Universita di Ferrara, Fossato
di Mortara, Italy)
J.K. Buolamwani (University of Tennessee,
Memphis, USA)
D.J. Canney (School of Pharmacy, Philadelphia,
PA, USA)
P. Chiba (Medizinischen Universität
Wien Raum, Währingerstraße, Austria)
B. Christensen (Alamo, USA)
S.B. Christensen (The Danish University of
Pharmaceutical Sciences, Copenhagen, Denmark)
M.J.C. Crabbe (University of Luton, Luton,
UK)
W-M. Dai (The Hong Kong University of Science
and Technology, Hong Kong SAR ,China)
R.B. de Alencastro (Institute de Quimica
da Universidade, RJ, Brazil)
Z. Debyser (Rega Institute for Medical Research,
Flanders, Belgium)
V.J. Demopoulos (University of Thessaloniki,
Thessaloniki ,Greece)
A.T. Dinkova-Kostova (Johns Hopkins University,
WBSB, USA)
S.W. Djuric (Abbott Laboratories, IL, USA)
J-M. Dogné (University of Liège
, Liège , Belgium)
G. Ecker (University of Vienna , Wien , Austria)
P. Englebienne (Biomedical Consultant, Zingem,
Belgium)
D. Fabbro (Novartis Pharma Inc., Basel, Switzerland)
P.M. Fischer (Discovery Research Cyclacel
Limited, Dundee ,Scotland)
D.M. Freymann (Northwestern University, Chicargo,
USA)
R. Gambari (Ferrara University, Ferrara,
Italy)
R.D. Gandour (Virginia Tech Blacksburg ,
VA , USA)
R.C. Gaudreault (CHUQ Hôpital Saint-François,
Québec, Canada)
T. Girbes (Universidad de Valladolid , Valladolid,
Spain)
R.A. Glennon (School of Medicine Virginia
Commonwealth , VA ,USA)
S. Goldstein (Institut de Recherches Servier,
Suresnes, France)
S. Guccione (University of Catania, Catania
, Italy)
A. Gueiffier (University of Tours, Tours,
France)
U. Haberkorn (University of Heidelberg Im
Neuenheimer, Heidelberg, Germany)
M.M. Harding (University of Sydney, NSW,
Australia)
A. Harvey (University of Strathclyde, Glasgow,
UK)
T. Högberg (7TM Pharma A/S Fremtidsvej
3, Hoersholm, Denmark)
J.F. Honek (University of Waterloo, Ontario,
Canada)
R.L. Hudkins (Medicinal Chemistry Cephalon,
Inc., PA ,USA)
P. Jackson (Johnson & Johnson Pharmaceutical
Research and Development L.L.C., Route, USA)
H.N. Jayaram (Indiana University School of
Medicine and Richard Roudebush VA Medical Center, IN, U.S.A.)
R. Jones (Arena Pharmaceuticals, CA, USA)
M. Jung (Yonsei University, Seoul, Korea)
M. Kahn (Institute For Chemical Genomics,
WA, USA)
M. Kassiou (Royal Prince Alfred Hospital,
Camperdown, Australia)
A.J. Kastin (Pennington Biomedical Research
Center, LA, USA)
J.F.W. Keana (University of Oregon, Eugene,
USA)
Y. Kiso (Kyoto Pharmaceutical University,
Kyoto, Japan)
K. Kuwano (Kyushu University, Fukooka, JAPAN)
D.J. Kyle (Purdue Pharma, Cranbury, USA)
P.Y. Lam (Bristol-Myers Squibb Co., Princeton,
USA)
M. Lee (Hope College, Holland, MI, USA)
C. Lee (National University of Singapore,
National Cancer Center, Singapore)
A. Mai (Università degli Studi di
Roma, Roma, Italy)
K. Maiese (Wayne State University School
of Medicine, MI, USA)
R. Mairs (Cancer Research UK Beatson Laboratories,
Glasgow, Scotland)
S. Malik (BioFrontiers Inc, WA, USA)
R. Mannhold (Heinrich-Heine-Universität,
Düsseldorf, Germany)
A.P. Marchand (University of North Texas,
NT, USA)
J.M.P. Martín (Universidad Autónoma
de Madrid, Madrid, Spain)
A. Martinez (Neuropharma Avda. de la Industria,
Madrid, Spain)
O.A. Mascaretti (University of Rosario Spinach,
Rosario, Argentina)
B. Masereel (University of Namur, Namur,
Belgium)
R.P. Mason (The University of Texas Southwestern,
Texas, USA)
G. Matarese (Università di Napoli
"Federico II", Napoli, Italy)
R. McGeary (The University of Queensland,
Queensland, Australia)
S. Mehta (Ambit Biosciences, CA, USA)
C. Meier (Universitaet Hamburg, Hamburg,
Germany)
J.J. Nestor, Jr. (Sequenom Pharmaceuticals,
CA, USA)
V.C.O. Njar (University of Maryland, MD,
USA)
F.G. Njoroge (Schering-Plough Research Institute,
New Jersy, USA)
M.H. Norman (Chemistry Research & Development
Amgen Inc., CA, USA)
I. Ojima (Institute of Chemical Biology &
Drug Discovery, NY, USA)
Y. Okada (Kobe Gauin University, Nishi-ku
Kobe, Japan)
D.W. Oliver (North-West University, Potchefstroom,
South Africa)
F. Ooms (Euroscreen S.A, Brussels ,Belgium
)
A.G. Papavassiliou (University of Athens,
Athens, Greece )
L.M. Pelus (Indiana University, Indiana,
USA)
G. Perry (University of Texas at San Antonio,
Texas 78249-0661, USA)
G. Poli (Vita-Salute San Raffaele University,
Milano, Italy)
P. Pourquier (Institut Bergonie & IECB,
Bordeaux cedex, France)
W. Priebe (The University of Texas M. D.
Anderson Cancer Center, Houston, TX, USA)
L. Prokai (University of Florida, FL, USA)
P.D. Roepe (Georgetown University, Washington
DC, USA)
V. Rotello (University of Massachusetts,
Amherst MA, USA)
S. Sarel (The Hebrew University of Jerusalem,
Jerusalem, Israel)
T.K. Sawyer (ARIAD Pharmaceuticals, Cambridge
MA, USA)
M. Searcey (University of East Anglia, Norwich
NR4 7TJ, UK)
R.P. Sharma (Molecular Biology School of
Biotical Sciences, Southampton, UK)
M.S. Sheikh (Upstate Medical University,
NY, USA)
R.D. Sindelar (The University of British
Columbia, Vancouver, Canada)
J.S. Skotnicki (Wyeth Research, NY, USA)
H. Stark (Institut fuer Pharmazeutische Chemie,
Frankfurt am Main, Germany)
N. Tagmatarchis (Universita di Trieste, Trieste,
Italy)
S. Takai (Osaka Medical College, Osaka, Japan)
K. Takeuchi (Lilly Research Laboratories
, IN, USA)
K. Takeuchi (Kyoto Pharmaceutical University,
Kyoto, Japan)
S.W. Topiol (Sandoz Research Institute, NJ,
USA)
N. Tuncel (Osmangazi University, Eskisehir,
Turkey)
H. Ulrich (Universidade de São Paulo,
S.P ,Brazil)
De-Y. Wang (The National University of Singapore,
Singapore)
D.J. Waxman (Boston University, MA , USA)
V. Weissig (Northeastern University, MA,
USA)
O. Werz (Institut für Pharmazeutische
Chemie, Frankfurt, Germany)
H.V. Wikstrom (University of Groningen A.
Deusinglaan 1, Groningen, Netherlands)
G. Willick (Institute for Biological Sciences,
ON , Canada , K1A 0R6)
Z. Xing (McMaster University, Ontario, Canada)
M. Yoshizumi (Nara Medical University School
of Medicine, Nara, Japan)
R. Zhang (University of Alabama at Birmingham,
USA)
F. Zunino (Istituto Nazionale Tumori, Milan,Italy)
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